Carbonic Anhydrase Inhibitors with Dual-Tail Moieties To Match the Hydrophobic and Hydrophilic Halves of the Carbonic Anhydrase Active Site-Reference-Cited by-同舟云学术

Carbonic Anhydrase Inhibitors with Dual-Tail Moieties To Match the Hydrophobic and Hydrophilic Halves of the Carbonic Anhydrase Active Site

Published:2015-01-27 Issue:3 Volume:58 Page:1494-1501
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tanpure Rajendra P.¹,Ren Bin²,Peat Thomas S.²,Bornaghi Laurent F.¹,Vullo Daniela³,Supuran Claudiu T.³,Poulsen Sally-Ann¹

Affiliation:

1. Eskitis Institute for Drug Discovery, Griffith University, Nathan, Queensland 4111, Australia

2. CSIRO, 343 Royal Parade, Parkville, Victoria 3052, Australia

3. Polo Scientifico, Neurofarba Department and Laboratorio di Chimica Bioinorganica, Università degli Studi di Firenze, Rm. 188, Via della Lastruccia 3, 50019 Sesto Fiorentino, Florence, Italy

Funder

European Commission

Australian Research Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm501798g

Reference36 articles.

1. New strategies for targeting the hypoxic tumour microenvironment in breast cancer

2. Hypoxia-induced carbonic anhydrase IX as a target for cancer therapy: From biology to clinical use

3. pH control mechanisms of tumor survival and growth

4. Interfering with pH regulation in tumours as a therapeutic strategy

5. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

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