Novel Organic Proteasome Inhibitors Identified by Virtual and in Vitro Screening-Reference-Cited by-同舟云学术

Novel Organic Proteasome Inhibitors Identified by Virtual and in Vitro Screening

Published:2009-11-17 Issue:1 Volume:53 Page:509-513
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Basse Nicolas¹,Montes Matthieu²,Maréchal Xavier¹,Qin Lixian¹,Bouvier-Durand Michelle¹,Genin Emilie³,Vidal Joëlle³,Villoutreix Bruno O.²,Reboud-Ravaux Michèle¹

Affiliation:

1. Enzymologie Moléculaire et Fonctionnelle, UR4, UPMC-Université de Paris 6, Case 256, 7 Quai Saint Bernard, F 75252 Paris Cedex 05, France

2. Inserm UMR-S 973, Molécules Thérapeutiques in Silico, Université Paris Diderot, 35 rue Hélène Brion, 75013 Paris, France

3. Chimie et Photonique Moléculaires, CNRS-UMR 6510, Université de Rennes 1, Campus Beaulieu, Bât. 10A, case 1012, CS 74205, 35042 Rennes Cedex, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9011092

Reference29 articles.

1. STRUCTURE AND FUNCTIONS OF THE 20S AND 26S PROTEASOMES

2. THE UBIQUITIN SYSTEM

3. The development of proteasome inhibitors as anticancer drugs

4. Proteasome Inhibitors in Cancer Therapy: Lessons from the First Decade

5. Proteasome Inhibition in the Treatment of Cancer

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