Structure-Based Design of High-Affinity and Selective Peptidomimetic Hepsin Inhibitors-Reference-Cited by-同舟云学术

Structure-Based Design of High-Affinity and Selective Peptidomimetic Hepsin Inhibitors

Published:2022-05-20 Issue:6 Volume:23 Page:2236-2242
ISSN:1525-7797
Container-title:Biomacromolecules
language:en
Short-container-title:Biomacromolecules

Author:

Knaff Philip Maximilian¹²,Müller Patrick³,Kersten Christian³^ORCID,Wettstein Lukas⁴,Münch Jan⁴^ORCID,Landfester Katharina¹^ORCID,Mailänder Volker¹²^ORCID

Affiliation:

1. Max Planck Institute for Polymer Research, Ackermannweg 10, Mainz 55128, Germany

2. Dermatology Clinic of the University Medicine of the Johannes Gutenberg University Mainz, Langenbeckstraße 1, Mainz 55131, Germany

3. Institute for Pharmaceutical and Biomedical Sciences, Johannes Gutenberg University Mainz, Staudingerweg 5, Mainz 55128, Germany

4. Institute of Molecular Virology, Ulm University Medical Center, Ulm 89081, Germany

Funder

Deutsche Forschungsgemeinschaft

Publisher

American Chemical Society (ACS)

Subject

Materials Chemistry,Polymers and Plastics,Biomaterials,Bioengineering

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.biomac.1c01011

Reference29 articles.

1. Kinases and Cancer

2. Cell surface–anchored serine proteases in cancer progression and metastasis

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4. Hepsin, a cell membrane-associated protease. Characterization, tissue distribution, and gene localization.

5. Hepsin is Highly Over Expressed in and a New Candidate for a Prognostic Indicator in Prostate Cancer

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