Insights into Actinium Complexes with Tetraacetates─AcBATA versus AcDOTA: Thermodynamic, Structural, and Labeling Properties

Author:

Matazova Ekaterina V.1ORCID,Egorova Bayirta V.1ORCID,Zubenko Anastasia D.2,Pashanova Anna V.23,Mitrofanov Artem A.1ORCID,Fedorova Olga A.23ORCID,Ermolaev Stanislav V.4,Vasiliev Aleksandr N.14,Kalmykov Stepan N.1

Affiliation:

1. Lomonosov Moscow State University, Leninskie Gory, 1/3, Moscow 119991, Russian Federation

2. A. N. Nesmeyanov Institute of Organoelement Compounds of Russian Academy of Sciences, Vavilova, 28, GSP-1, Moscow 119334, Russian Federation

3. Mendeleev University of Chemistry and Technology of Russia, Miusskaya sqr., 9, Moscow 125047, Russian Federation

4. Institute for Nuclear Research of Russian Academy of Sciences, 60th October Anniversary Prospect, 7a, Moscow 117312, Russian Federation

Funder

Russian Science Foundation

Publisher

American Chemical Society (ACS)

Subject

Inorganic Chemistry,Physical and Theoretical Chemistry

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3. “ FDA Letter of Approval for LUTATHERA”, can be found under https://www.accessdata.fda.gov/drugsatfda_docs/appletter/2018/208700Orig1s000ltr.pdf (accessed April 23, 2019).

4. “ FDA Letter of Approval for PLUVICTO”, can be found under https://www.accessdata.fda.gov/drugsatfda_docs/label/2022/215833s000lbl.pdf (accessed on March 23, 2022).

5. DNA Double Strand Breaks as Predictor of Efficacy of the Alpha-Particle Emitter Ac-225 and the Electron Emitter Lu-177 for Somatostatin Receptor Targeted Radiotherapy

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