3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A New Scaffold for the Selective Inhibition of Monoamine Oxidase B-Reference-Cited by-同舟云学术

3-Acetyl-2,5-diaryl-2,3-dihydro-1,3,4-oxadiazoles: A New Scaffold for the Selective Inhibition of Monoamine Oxidase B

Published:2011-08-17 Issue:18 Volume:54 Page:6394-6398
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Maccioni Elias¹,Alcaro Stefano²,Cirilli Roberto³,Vigo Sara¹,Cardia Maria Cristina¹,Sanna Maria Luisa¹,Meleddu Rita¹,Yanez Matilde⁴,Costa Giosuè²,Casu Laura¹,Matyus Peter⁵,Distinto Simona²

Affiliation:

1. Dipartimento Farmaco Chimico Tecnologico, University of Cagliari, Via Ospedale 72, 09124, Cagliari, Italy

2. Dipartimento di Scienze Farmacobiologiche, University “Magna Græcia” di Catanzaro, Complesso “Ninì Barbieri”, 88021 Roccelletta di Borgia (CZ), Italy

3. Dipartimento del Farmaco, Istituto Superiore di Sanità, V. le Regina Elena 299, 00161 Roma, Italy

4. Departamento de Farmacología and Instituto de Farmacia Industrial, Universidad de Santiago de Compostela, Campus Universitario Sur, E-15782 Santiago de Compostela, Spain

5. Department of Organic Chemistry, Semmelweis University; Högyes E. u. 7, H-1092 Budapest, Hungary

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm2002876

Reference23 articles.

1. The therapeutic potential of monoamine oxidase inhibitors

2. The increasing role of monoamine oxidase type B inhibitors in Parkinson's disease therapy

3. Increased monoamine oxidase b activity in plaque-associated astrocytes of Alzheimer brains revealed by quantitative enzyme radioautography

4. Oxidative α-Ketoglutarate Dehydrogenase Inhibition via Subtle Elevations in Monoamine Oxidase B Levels Results in Loss of Spare Respiratory Capacity

5. Comprehensive review of rasagiline, a second-generation monoamine oxidase inhibitor, for the treatment of Parkinson's Disease

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