Striking Effect of Hydroxamic Acid Substitution on the Phosphodiesterase Type 4 (PDE4) and TNFα Inhibitory Activity of Two Series of Rolipram Analogues: Implications for a New Active Site Model of PDE4
Author:
Affiliation:
1. Central Research Division, Pfizer Inc., Groton, Connecticut 06340
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm970685m
Reference22 articles.
1. Phosphodiesterase inhibitors: new opportunities for the treatment of asthma.
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