On-Bead Screening of a Combinatorial Fumaric Acid Derived Peptide Library Yields Antiplasmodial Cysteine Protease Inhibitors with Unusual Peptide Sequences-Reference-Cited by-同舟云学术

On-Bead Screening of a Combinatorial Fumaric Acid Derived Peptide Library Yields Antiplasmodial Cysteine Protease Inhibitors with Unusual Peptide Sequences

Published:2009-08-31 Issue:18 Volume:52 Page:5662-5672
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Machon Uwe¹,Büchold Christian²,Stempka Martin²,Schirmeister Tanja²,Gelhaus Christoph³,Leippe Matthias³,Gut Jiri⁴,Rosenthal Philip J.⁴,Kisker Caroline⁵,Leyh Matthias⁵,Schmuck Carsten¹

Affiliation:

1. Institute of Organic Chemistry, University of Duisburg-Essen, Universitätstrasse 7, 45141 Essen, Germany

2. Institute of Pharmacy and Food Chemistry, University of Würzburg, Am Hubland, 97074 Würzburg, Germany

3. Institute of Zoology, University of Kiel, Olshausenstrasse 40, 24098 Kiel, Germany

4. Department of Medicine, San Francisco General Hospital, University of California, San Francisco, Box 0811, San Francisco, California 94143

5. Rudolf-Virchow-Zentrum DFG-Forschungszentrum für Experimentelle Biomedizin, Versbacher Strasse 9, 97078 Würzburg, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm900629w

Reference75 articles.

1. Human African trypanosomiasis: clinical presentation and immune response

2. Cysteine Proteinases of Trypanosome Parasites Novel Targets for Chemotherapy

3. Chemotherapeutic Agents Against Malaria: What Next After Chloroquine?

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