Discovery of 4,4-Disubstituted Quinazolin-2-ones as T-Type Calcium Channel Antagonists
Author:
Affiliation:
1. Departments of Medicinal Chemistry
2. Drug Metabolism and Pharmacokinetics
3. Depression and Circadian Disorders
4. Parkinson's Disease
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/ml100004r
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1. Nomenclature of Voltage-Gated Calcium Channels
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3. Differential Distribution of Three Members of a Gene Family Encoding Low Voltage-Activated (T-Type) Calcium Channels
4. Discovery and main pharmacological properties of mibefradil (Ro 40-5967), the first selective T-type calcium channel blocker
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