Small Molecule Inhibitors of Bacillus anthracis Protective Antigen Proteolytic Activation and Oligomerization-Reference-Cited by-同舟云学术

Small Molecule Inhibitors of Bacillus anthracis Protective Antigen Proteolytic Activation and Oligomerization

Published:2012-09-18 Issue:18 Volume:55 Page:7998-8006
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Wein Alexander N.¹,Williams Brian N.¹,Liu Shihui¹,Ermolinsky Boris²,Provenzano Daniele²,Abagyan Ruben³,Orry Andrew⁴,Leppla Stephen H.¹,Peredelchuk Michael²

Affiliation:

1. Microbial Pathogenesis Section, Laboratory of Parasitic Diseases, National Institute of Allergy and Infectious Diseases, National Institutes of Health, 33 North Drive, Bethesda, Maryland 20892, United States

2. Department of Biomedical Sciences, University of Texas Brownsville, 80 Fort Brown, Brownsville, Texas 78520, United States

3. Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California—San Diego, 9500 Gilman Drive, La Jolla, California 92093, United States

4. MolSoft LLC, 11199 Sorrento Valley Road S209, San Diego, California 92121, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300804e

Reference70 articles.

1. Pathophysiology of anthrax

2. The Protective Antigen Component of Anthrax Toxin Forms Functional Octameric Complexes

3. Cellular and systemic effects of anthrax lethal toxin and edema toxin

4. Bacillus anthracis physiology and genetics

5. Anthrax Toxin Targeting of Myeloid Cells through the CMG2 Receptor Is Essential for Establishment of Bacillus anthracis Infections in Mice

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