Design, Synthesis, and Dopamine Receptor Modulating Activity of Spiro Bicyclic Peptidomimetics of l-Prolyl-l-leucyl-glycinamide-Reference-Cited by-同舟云学术

Design, Synthesis, and Dopamine Receptor Modulating Activity of Spiro Bicyclic Peptidomimetics of l-Prolyl-l-leucyl-glycinamide

Published:1999-01-29 Issue:4 Volume:42 Page:628-637
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Khalil Ehab M.¹,Ojala William H.¹,Pradhan Ashish¹,Nair Venugopalan D.¹,Gleason William B.¹,Mishra Ram K.¹,Johnson Rodney L.¹

Affiliation:

1. Department of Medicinal Chemistry and The Biomedical Engineering Center and Department of Laboratory Medicine and Pathology, University of Minnesota, Minneapolis, Minnesota 55455, and Department of Psychiatry and Behavioural Neuroscience, McMaster University, Hamilton, Ontario L8N 3Z5, Canada

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm980525q

Reference29 articles.

1. Effect of L-prolyl-L-leucyl-glycinamide (PLG) on neuroleptic-induced catalepsy and dopamine/neuroleptic receptor bindings

2. Interaction of l-Prolyl-l-Leucyl Glycinamide with Dopamine D2Receptor: Evidence for Modulation of Agonist Affinity States in Bovine Striatal Membranes

3. Modulation of high-affinity CNS dopamine D2 receptor by l-pro-l-leu-glycinamide (PLG) analogue

4. Design, Synthesis, X-ray Analysis, and Dopamine Receptor-Modulating Activity of Mimics of the "C5" Hydrogen-Bonded Conformation in the Peptidomimetic 2-Oxo-3(R)-[(2(S)-pyrrolidinylcarbonyl)amino]-1-pyrrolidineacetamide

5. Design, Synthesis, and Dopamine Receptor Modulating Activity of Diketopiperazine Peptidomimetics of l-Prolyl-l-leucylglycinamide

Cited by 65 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Structure-based design of novel melanin-concentrating hormone receptor-1 ligands based on saturated nitrogen-containing heterocycles;Bioorganic & Medicinal Chemistry Letters;2023-03

2. Allosteric Modulators of Dopamine D2 Receptors for Fine-Tuning of Dopaminergic Neurotransmission in CNS Diseases: Overview, Pharmacology, Structural Aspects and Synthesis;Molecules;2022-12-25

3. Pseudoprolines as stereoelectronically tunable proline isosteres;Bioorganic & Medicinal Chemistry Letters;2022-11

4. Peptidomimetics: An Overview of Recent Medicinal Chemistry Efforts toward the Discovery of Novel Small Molecule Inhibitors;Journal of Medicinal Chemistry;2022-05-23

5. New Methods for the Synthesis of Spirocyclic Cephalosporin Analogues;Molecules;2021-10-05