The Process Development of Ravuconazole: An Efficient Multikilogram Scale Preparation of an Antifungal Agent-Reference-Cited by-同舟云学术

The Process Development of Ravuconazole: An Efficient Multikilogram Scale Preparation of an Antifungal Agent

Published:2009-07-17 Issue:4 Volume:13 Page:716-728
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Pesti Jaan¹,Chen Chien-Kuang¹,Spangler Lori¹,DelMonte Albert J.¹,Benoit Serge¹,Berglund Derek¹,Bien Jeffrey¹,Brodfuehrer Paul¹,Chan Yeung¹,Corbett Elisabeth¹,Costello Carrie¹,DeMena Paul¹,Discordia Robert P.¹,Doubleday Wendel¹,Gao Zhinong¹,Gingras Stephane¹,Grosso John¹,Haas Oscar¹,Kacsur David¹,Lai Chiajen¹,Leung Simon¹,Miller Melanie¹,Muslehiddinoglu Jale¹,Nguyen Nina¹,Qiu Jun¹,Olzog Martina¹,Reiff Emily¹,Thoraval Dominique¹,Totleben Michael¹,Vanyo Dale¹,Vemishetti Purushotham¹,Wasylak John¹,Wei Chenkou¹

Affiliation:

1. Process Research and Development, Bristol-Myers Squibb Pharmaceutical Co., One Squibb Drive, P.O. Box 191, New Brunswick, New Jersey, 08903-0191, U.S.A.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op900065c

Reference85 articles.

1. Aspects of this work were also carried out at Bristol-Myers Squibb’s facilities in Princeton, NJ; Candiac, Canada; and Syracuse, NY.

2. Ravuconazole was licensed from Eisai Co. Ltd. References to earlier studies include:

3. In vitro and in vivo antifungal activities of ER-30346, a novel oral triazole with a broad antifungal spectrum

4. In Vitro Activity of a New Oral Triazole, BMS-207147 (ER-30346)

Cited by 43 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Exploring triazole-based drugs: Synthesis, application, FDA approvals, and clinical trial updates–A comprehensive review;Tetrahedron;2024-08

2. The immobilization of L-Valine on superparamagnetic Fe ₃ O ₄ nanoparticles as a novel, recoverable and green nanocatalyst for the synthesis of new thiazole derivatives;Journal of Sulfur Chemistry;2024-07-24

3. Use of Impinging Jet to Improve Scalability in the Preparation of the ABBV-154 Drug-Linker;Organic Process Research & Development;2024-06-28

4. Discovery of a Novel Potent Tetrazole Antifungal Candidate with High Selectivity and Broad Spectrum;Journal of Medicinal Chemistry;2024-04-10

5. Asymmetric Synthesis of Triazole Antifungal Agents Enabled by an Upgraded Strategy for the Key Epoxide Intermediate;The Journal of Organic Chemistry;2024-03-21