Synthesis and Evaluation of Isomeric (17α,20E)-11β-Methoxy-21-(trifluoromethylphenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17β-diols as ERα-Hormone Binding Domain Ligands: Effect of the Methoxy Group on Receptor Binding and Uterotrophic Growth-Reference-Cited by-同舟云学术

Synthesis and Evaluation of Isomeric (17α,20E)-11β-Methoxy-21-(trifluoromethylphenyl)-19-norpregna-1,3,5(10),20-tetraene-3,17β-diols as ERα-Hormone Binding Domain Ligands: Effect of the Methoxy Group on Receptor Binding and Uterotrophic Growth

Published:2007-01-09 Issue:3 Volume:50 Page:472-479
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hanson Robert N.¹,Tongcharoensirikul Pakamas¹,Dilis Robert¹,Hughes Alun¹,DeSombre Eugene R.¹

Affiliation:

1. Department of Chemistry and Chemical Biology, Northeastern University, 360 Huntington Avenue, Boston, Massachusetts 02115, and The Ben May Institute for Cancer Research, The University of Chicago, 5841 South Maryland Avenue, Chicago, Illinois 60637

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060940f

Reference53 articles.

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