(±)-(1S,2R,5S)-5-Amino-2-fluorocyclohex-3-enecarboxylic Acid. A Potent GABA Aminotransferase Inactivator that Irreversibly Inhibits via an Elimination−Aromatization Pathway-Reference-Cited by-同舟云学术

(±)-(1S,2R,5S)-5-Amino-2-fluorocyclohex-3-enecarboxylic Acid. A Potent GABA Aminotransferase Inactivator that Irreversibly Inhibits via an Elimination−Aromatization Pathway

Published:2006-11-08 Issue:48 Volume:45 Page:14513-14522
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Wang Zhiyong¹,Yuan Hai¹,Nikolic Dejan¹,Van Breemen Richard B.¹,Silverman Richard B.¹

Affiliation:

1. Department of Chemistry, Department of Biochemistry, Molecular Biology, and Cell Biology, and Center for Drug Discovery and Chemical Biology, Northwestern University, Evanston, Illinois 60208-3113, and Department of Medicinal Chemistry and Pharmacognosy, University of Illinois, Chicago, Illinois 60612-7231

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/bi061592m

Reference43 articles.

1. Chemical Nature of Synaptic Transmission in Vertebrates

2. GABA in Epilepsy: The Pharmacologic Basis

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