Preliminary Structure–Activity Relationships and Biological Evaluation of Novel Antitubercular Indolecarboxamide Derivatives Against Drug-Susceptible and Drug-Resistant Mycobacterium tuberculosis Strains-Reference-Cited by-同舟云学术

Preliminary Structure–Activity Relationships and Biological Evaluation of Novel Antitubercular Indolecarboxamide Derivatives Against Drug-Susceptible and Drug-Resistant Mycobacterium tuberculosis Strains

Published:2013-05-03 Issue:10 Volume:56 Page:4093-4103
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Onajole Oluseye K.¹,Pieroni Marco¹,Tipparaju Suresh K.¹,Lun Shichun²,Stec Jozef¹,Chen Gang¹,Gunosewoyo Hendra¹,Guo Haidan²,Ammerman Nicole C.²³,Bishai William R.²³⁴,Kozikowski Alan P.¹

Affiliation:

1. Department of Medicinal Chemistry and Pharmacognosy, College of Pharmacy, University of Illinois at Chicago, 833 South Wood Street, Chicago, Illinois 60612, United States

2. Center for Tuberculosis Research, Department of Medicine, Division of Infectious Disease, Johns Hopkins School of Medicine, Baltimore, Maryland 21231-1044, United States

3. KwaZulu-Natal Research Institute for Tuberculosis and HIV, Nelson R. Mandela School of Medicine, 719 Umbilo Road, Durban 4001, KwaZulu-Natal, South Africa

4. Howard Hughes Medical Institute, 4000 Jones Bridge Road, Chevy Chase, Maryland 20815-6789, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm4003878

Reference32 articles.

1. Tuberculosis;Fact Sheet no. 104;World Health Organisation:Geneva, 2013; http://www.who.int/mediacentre/factsheets/fs104/en/index.html(accessed February 11, 2013).

2. Global Tuberculosis Report 2012;World Health Organisation:Geneva, 2012; http://apps.who.int/iris/bitstream/10665/75938/1/9789241564502_eng.pdf(accessed January 8, 2013).

3. Directly observed therapy (DOT) for tuberculosis: why, when, how and if?

4. Epidemiology and Challenges to the Elimination of Global Tuberculosis

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