1. Chemical Biology and Organic Chemistry, Bijvoet Center for Biomolecular Research, Utrecht University, Padualaan 8, 3584 CH Utrecht, The Netherlands, Medicinal Chemistry and Chemical Biology, Utrecht Institute for Pharmaceutical Sciences, Utrecht University, Sorbonnelaan 16, 3584 CA Utrecht, The Netherlands, Centro de Química-Física Molecular, Complexo Interdisciplinar, Instituto Superior Técnico, Av. Rovisco Pais, 1049-001 Lisbon, Portugal, Faculdade de Farmácia da Universidade de Coimbra, 3000-295...