Affinity Crystallography: A New Approach to Extracting High-Affinity Enzyme Inhibitors from Natural Extracts

Author:

Aguda Adeleke H.1,Lavallee Vincent1,Cheng Ping1,Bott Tina M.1,Meimetis Labros G.1,Law Simon1,Nguyen Nham T.1,Williams David E.1,Kaleta Jadwiga1,Villanueva Ivan1,Davies Julian1,Andersen Raymond J.1,Brayer Gary D.1,Brömme Dieter1

Affiliation:

1. Department of Oral Biological and Medical Sciences, Faculty of Dentistry, ‡Department of Biochemistry and Molecular Biology, Faculty of Medicine, §Department of Chemistry and Earth, Ocean & Atmospheric Sciences, Faculty of Science, ⊥Department of Microbiology, Faculty of Science, and ∥Centre for Blood Research, University of British Columbia, Vancouver, BC Canada, V6T 1Z3

Funder

Canadian Institutes of Health Research

Institute of Musculoskeletal Health and Arthritis

Natural Sciences and Engineering Research Council of Canada

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Complementary and alternative medicine,Drug Discovery,Pharmaceutical Science,Pharmacology,Molecular Medicine,Analytical Chemistry

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