Design, Synthesis, and Pharmacological Evaluation of Pyridinic Analogues of Nimesulide as Cyclooxygenase-2 Selective Inhibitors-Reference-Cited by-同舟云学术

Design, Synthesis, and Pharmacological Evaluation of Pyridinic Analogues of Nimesulide as Cyclooxygenase-2 Selective Inhibitors

Published:2004-12-01 Issue:27 Volume:47 Page:6749-6759
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Julémont Fabien¹,de Leval Xavier¹,Michaux Catherine¹,Renard Jean-François¹,Winum Jean-Yves¹,Montero Jean-Louis¹,Damas Jacques¹,Dogné Jean-Michel¹,Pirotte Bernard¹

Affiliation:

1. Natural and Synthetic Drugs Research Centre, Laboratory of Medicinal Chemistry, Université de Liège, 1, Avenue de l'Hôpital, B36, B-4000 Liège, Belgium, Department of Molecular and Structural Chemistry, Université de Namur, 61, Rue de Bruxelles, B-5000 Namur, Belgium, Laboratoire de Chimie Biomoléculaire, Université Montpellier II, UMR 5032, ENSCM, 8, Rue de l'Ecole Normale, 34296 Montpellier Cedex, France, and Department of Human Physiology, Université de Liège, 1, Avenue de l'Hôpital, B23, B-4000 Liège...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049480l

Reference39 articles.

1. Cyclooxygenases: Structural, Cellular, and Molecular Biology

2. Cyclooxygenase-1 and -2 expression in rheumatoid synovial tissues. Effects of interleukin-1 beta, phorbol ester, and corticosteroids.

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