Discovery and Labeling of High-Affinity 3,4-Diarylpyrazolines as Candidate Radioligands for In Vivo Imaging of Cannabinoid Subtype-1 (CB1) Receptors-Reference-Cited by-同舟云学术

Discovery and Labeling of High-Affinity 3,4-Diarylpyrazolines as Candidate Radioligands for In Vivo Imaging of Cannabinoid Subtype-1 (CB1) Receptors

Published:2008-08-28 Issue:18 Volume:51 Page:5608-5616
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Donohue Sean R.¹,Pike Victor W.¹,Finnema Sjoerd J.¹,Truong Phong¹,Andersson Jan¹,Gulyás Balázs¹,Halldin Christer¹

Affiliation:

1. Molecular Imaging Branch, National Institute of Mental Health, National Institutes of Health, Bethesda, Maryland 20892, Karolinska Institutet, Department of Clinical Neuroscience, Psychiatry Section, Karolinska Hospital, S-17176 Stockholm, Sweden

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800329z

Reference46 articles.

1. Review of Cannabinoids and their Antiemetic Effectiveness

2. CANNABINOID RECEPTORS AS THERAPEUTIC TARGETS

3. The Endocannabinoid System: Drug Targets, Lead Compounds, and Potential Therapeutic Applications

4. Cannabinoids and the Digestive Tract

5. Delta-9-tetrahydrocannabinol differentially suppresses emesis versus enhanced locomotor activity produced by chemically diverse dopamine D/D receptor agonists in the least shrew ()

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