Synthesis, Inhibitory Activity of Cholinesterases, and Neuroprotective Profile of Novel 1,8-Naphthyridine Derivatives-Reference-Cited by-同舟云学术

Synthesis, Inhibitory Activity of Cholinesterases, and Neuroprotective Profile of Novel 1,8-Naphthyridine Derivatives

Published:2010-06-24 Issue:14 Volume:53 Page:5129-5143
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

de los Ríos Cristóbal¹²³,Egea Javier¹,Marco-Contelles José²,León Rafael¹,Samadi Abdelouahid²,Iriepa Isabel³,Moraleda Ignacio³,Gálvez Enrique³,García Antonio G.¹⁴,López Manuela G.¹,Villarroya Mercedes¹,Romero Alejandro¹

Affiliation:

1. Departamento de Farmacología y Terapéutica, Facultad de Medicina, Instituto Teófilo Hernando, Universidad Autónoma de Madrid, C/Arzobispo Morcillo 4, 28029 Madrid, Spain

2. Laboratorio de Radicales Libres y Química Computacional, Instituto de Química Orgánica General, Consejo Superior de Investigaciones Científicas, C/Juan de la Cierva 3, 28006 Madrid, Spain

3. Departamento de Química Orgánica, Facultad de Farmacia, Universidad de Alcalá de Henares, Ctra. Barcelona, Km. 33.5, 28817, Alcalá de Henares, Spain

4. Servicio de Farmacología Clínica, Hospital Universitario de la Princesa, C/Diego de León 62, 28006 Madrid, Spain

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm901902w

Reference74 articles.

1. A Century of Alzheimer's Disease

2. Targeting Beta-Amyloid Pathogenesis Through Acetylcholinesterase Inhibitors

3. Hyperphosphorylation of Microtubule-Associated Protein Tau: A Promising Therapeutic Target for Alzheimer Disease

4. Evidence of Oxidative Stress in Alzheimer's Disease Brain and Antioxidant Therapy

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