Identification of a Nonpeptidic and Conformationally Restricted Bradykinin B1 Receptor Antagonist with Anti-Inflammatory Activity-Reference-Cited by-同舟云学术

Identification of a Nonpeptidic and Conformationally Restricted Bradykinin B1 Receptor Antagonist with Anti-Inflammatory Activity

Published:2007-01-23 Issue:4 Volume:50 Page:607-610
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

D'Amico Derin C.¹,Aya Toshi¹,Human Jason¹,Fotsch Christopher¹,Chen Jian Jeffrey¹,Biswas Kaustav¹,Riahi Bobby¹,Norman Mark H.¹,Willoughby Christopher A.¹,Hungate Randall¹,Reider Paul J.¹,Biddlecome Gloria¹,Lester-Zeiner Dianna¹,Van Staden Carlo¹,Johnson Eileen¹,Kamassah Augustus¹,Arik Leyla¹,Wang Judy¹,Viswanadhan Vellarkad N.¹,Groneberg Robert D.¹,Zhan James¹,Suzuki Hideo¹,Toro Andras¹,Mareska David A.¹,Clarke David E.¹,Harvey Darren M.¹,Burgess Laurence E.¹,Laird Ellen R.¹,Askew Benny¹,Ng Gordon¹

Affiliation:

1. Chemistry Research and Development, Neuroscience, HTS/Molecular Pharmacology, Molecular Structure and Design, and Inflammation, Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, and Array BioPharma, 3200 Walnut Street, Boulder, Colorado 80301

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm061224g

Reference19 articles.

1. Bradykinin and inflammatory pain

2. Kinin Formation: Mechanisms and Role in Inflammatory Disorders

3. Cardiovascular effects of peptide kinin B2 receptor antagonists in rats

4. Cardiovascular effects of peptide kinin B2 receptor antagonists in rats

5. Hypoalgesia and altered inflammatory responses in mice lacking kinin B1 receptors

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