Comparison of the Permeability of Metoprolol and Labetalol in Rat, Mouse, and Caco-2 Cells: Use as a Reference Standard for BCS Classification-Reference-Cited by-同舟云学术

Comparison of the Permeability of Metoprolol and Labetalol in Rat, Mouse, and Caco-2 Cells: Use as a Reference Standard for BCS Classification

Published:2013-02-04 Issue:3 Volume:10 Page:958-966
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Incecayir Tuba¹²,Tsume Yasuhiro¹,Amidon Gordon L.¹

Affiliation:

1. Department of Pharmaceutical Sciences, College of Pharmacy, University of Michigan, Ann Arbor, Michigan 48109-1065, United States

2. Department of Pharmaceutical Technology, Faculty of Pharmacy, Gazi University, Ankara 06330, Turkey

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/mp300410n

Reference51 articles.

1. U.S. Food and Drug Administration, Center for Drug Evaluationand Research (CDER). Guidance for Industry: Bioavailability and BioequivalenceStudies for Orally Administered Drug Products—General Considerations,March (2003; Division of Drug Information Branch, HFD-240,Center for Drug Evaluation and Research, FDA:Rockville, MD;http://www.fda.gov/downloads/Drugs/GuidanceComplianceRegulatoryInformation/Guidances/UCM070124.pdf.

2. European Medicines Agency (EMEA) Committeefor MedicinalProducts for Human Use. Guideline on the Investigation of Bioequivalence;Doc.Ref.: CPMP/EWP/QWP/1401/98Rev.1/Corr; EMEA:London, January 20, 2010; http://www.emea.europa.eu/docs/en_GB/document_library/Scientific_guideline/2010/01/WC500070039.pdf.

3. Summary Workshop Report: Bioequivalence, Biopharmaceutics Classification System, and Beyond

4. The BCS, BDDCS, and Regulatory Guidances

Cited by 68 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A 3D in-vitro biomimicking Caco-2 intestinal permeability model-based assessment of physically modified telmisartan towards an alkalizer-free formulation development;European Journal of Pharmaceutics and Biopharmaceutics;2024-10

2. Studies on pharmacokinetic properties and intestinal absorption mechanism of sanguinarine chloride: in vivo and in situ;Toxicology Mechanisms and Methods;2024-08

3. Biowaiver Monograph for Immediate-Release Solid Oral Dosage Forms: Raltegravir Potassium;Journal of Pharmaceutical Sciences;2024-08

4. In silico, in situ, in vitro, and in vivo predictive methods for modeling formulation performance;From Current to Future Trends in Pharmaceutical Technology;2024

5. Challenges in Permeability Assessment for Oral Drug Product Development;Pharmaceutics;2023-09-28