1-Alkyl-benzotriazole-5-carboxylic Acids Are Highly Selective Agonists of the Human Orphan G-Protein-Coupled Receptor GPR109b-Reference-Cited by-同舟云学术

1-Alkyl-benzotriazole-5-carboxylic Acids Are Highly Selective Agonists of the Human Orphan G-Protein-Coupled Receptor GPR109b

Published:2006-01-24 Issue:4 Volume:49 Page:1227-1230
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Semple Graeme¹,Skinner Philip J.¹,Cherrier Martin C.¹,Webb Peter J.¹,Sage Carleton R.¹,Tamura Susan Y.¹,Chen Ruoping¹,Richman Jeremy G.¹,Connolly Daniel T.¹

Affiliation:

1. Medicinal Chemistry and Discovery Biology, Arena Pharmaceuticals, 6166 Nancy Ridge Drive, San Diego, California 92121

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm051099t

Reference10 articles.

1. Influence of nicotinic acid on serum cholesterol in man

2. Characterization of a G Protein-Coupled Receptor for Nicotinic Acid

3. Molecular Identification of High and Low Affinity Receptors for Nicotinic Acid

4. Molecular identification of nicotinic acid receptor

5. PUMA-G and HM74 are receptors for nicotinic acid and mediate its anti-lipolytic effect

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