Metal Impurities Cause False Positives in High-Throughput Screening Campaigns
Author:
Affiliation:
1. Discovery Chemistry, ‡Discovery Technologies, and §Inflammation Discovery, Roche pRED, 340 Kingsland Street, Nutley, New Jersey 07110, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/ml3003296
Reference35 articles.
1. Education reforms struggle against apartheid's legacy
2. The application of high-throughput screening to novel lead discovery
3. High-throughput screening: new technology for the 21st century
4. NMR-Based Quality Control Approach for the Identification of False Positives and False Negatives in High Throughput Screening
5. Learning from the Data: Mining of Large High-Throughput Screening Databases
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