Combination of Molecular Modeling, Site-Directed Mutagenesis, and SAR Studies To Delineate the Binding Site of Pyridopyrimidine Antagonists on the Human CCK1 Receptor-Reference-Cited by-同舟云学术

Combination of Molecular Modeling, Site-Directed Mutagenesis, and SAR Studies To Delineate the Binding Site of Pyridopyrimidine Antagonists on the Human CCK1 Receptor

Published:2005-07-01 Issue:15 Volume:48 Page:4842-4850
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Martín-Martínez Mercedes¹,Marty Anne¹,Jourdan Maud¹,Escrieut Chantal¹,Archer Elodie¹,González-Muñiz Rosario¹,García-López M. Teresa¹,Maigret Bernard¹,Herranz Rosario¹,Fourmy Daniel¹

Affiliation:

1. Instituto de Química Médica (CSIC), Juan de la Cierva 3, E-28006 Madrid, Spain, INSERM U 531, Institut Louis Bugnard, TSA 50032, CHU Rangueil, Bat. L3, 31059 Toulouse Cedex 9, France, and Laboratoire de Chimie Théorique, UMR CNRS Université de Nancy, 54506 Vandoeuvre les Nancy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0501127

Reference41 articles.

1. Cholecystokinin and regulation of pancreatic acinar cell function

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