Synthesis and Antibacterial Activity of a Novel Series of Potent DNA Gyrase Inhibitors. Pyrazole Derivatives-Reference-Cited by-同舟云学术

Synthesis and Antibacterial Activity of a Novel Series of Potent DNA Gyrase Inhibitors. Pyrazole Derivatives

Published:2004-06-05 Issue:14 Volume:47 Page:3693-3696
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tanitame Akihiko¹,Oyamada Yoshihiro¹,Ofuji Keiko¹,Fujimoto Mika¹,Iwai Noritaka¹,Hiyama Yoichi¹,Suzuki Kenji¹,Ito Hideaki¹,Terauchi Hideo¹,Kawasaki Motoji¹,Nagai Kazuo¹,Wachi Masaaki¹,Yamagishi Jun-ichi¹

Affiliation:

1. Chemistry Research Laboratories, Pharmacology and Microbiology Research Laboratories, Dainippon Pharmaceutical Co., Ltd., 33-94, Enoki, Suita, Osaka 564-0053, Japan, Department of Bioengineering, Tokyo Institute of Technology, 4259, Nagatsuda, Midori-ku, Yokohama 226-8501, Japan, and Department of Biological Chemistry, Chubu University, 1200 Matsumoto, Kasugai, Aichi 487-8501, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030394f

Reference9 articles.

1. Cloning and primary structure of Staphylococcus aureus DNA topoisomerase IV: a primary target of fluoroquinolones

2. Pyridonecarboxylic acids as antibacterial agents. Part 14. Synthesis and structure-activity relationships of 5-substituted 6,8-difluoroquinolones, including sparfloxacin, a new quinolone antibacterial agent with improved potency

3. The interaction between coumarin drugs and DNA gyrase

4. Novel Inhibitors of DNA Gyrase: 3D Structure Based Biased Needle Screening, Hit Validation by Biophysical Methods, and 3D Guided Optimization. A Promising Alternative to Random Screening

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