Novel N-Substituted Indol-3-ylglyoxylamides Probing the LDi and L1/L2 Lipophilic Regions of the Benzodiazepine Receptor Site in Search for Subtype-Selective Ligands-Reference-Cited by-同舟云学术

Novel N-Substituted Indol-3-ylglyoxylamides Probing the LDi and L1/L2 Lipophilic Regions of the Benzodiazepine Receptor Site in Search for Subtype-Selective Ligands

Published:2007-03-03 Issue:7 Volume:50 Page:1627-1634
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Primofiore Giampaolo¹,Taliani Sabrina¹,Da Settimo Federico¹,Marini Anna Maria¹,La Motta Concettina¹,Simorini Francesca¹,Patrizi Maria Paola¹,Sergianni Valentina¹,Novellino Ettore¹,Greco Giovanni¹,Cosimelli Barbara¹,Calderone Vincenzo¹,Montali Marina¹,Besnard François¹,Martini Claudia¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy, Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli “Federico II”, Via Domenico Montesano, 49, 80131 Napoli, Italy, Department of Molecular and Functional Genomics, Synthélabo, 10 rue des Carrières, 92500 Rueil-Malmaison, France, and Dipartimento di Psichiatria, Neurobiologia, Farmacologia e Biotecnologie, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0607707

Reference37 articles.

1. GABA-Activated Ligand Gated Ion Channels: Medicinal Chemistry and Molecular Biology

2. An update on GABAA receptors

3. Mapping of the Benzodiazepine Recognition Site on GABA-A Receptors

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