4-Benzyl and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones: In Vitro Evaluation of New C-3-Amino-Substituted and C-5,6-Alkyl-Substituted Analogues against Clinically Important HIV Mutant Strains-Reference-Cited by-同舟云学术

4-Benzyl and 4-Benzoyl-3-dimethylaminopyridin-2(1H)-ones: In Vitro Evaluation of New C-3-Amino-Substituted and C-5,6-Alkyl-Substituted Analogues against Clinically Important HIV Mutant Strains

Published:2005-02-08 Issue:6 Volume:48 Page:1948-1964
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Benjahad Abdellah¹,Croisy Martine¹,Monneret Claude¹,Bisagni Emile¹,Mabire Dominique¹,Coupa Sophie¹,Poncelet Alain¹,Csoka Imre¹,Guillemont Jérôme¹,Meyer Christophe¹,Andries Koen¹,Pauwels Rudi¹,de Béthune Marie-Pierre¹,Himmel Daniel M.¹,Das Kalyan¹,Arnold Eddy¹,Nguyen Chi Hung¹,Grierson David S.¹

Affiliation:

1. Laboratoire de Pharmacochimie, Section de Recherche, UMR 176 CNRS-Institut Curie, Batiment 110, Centre Universitaire, 91405 Orsay, France, Medicinal Chemistry Department, Johnson & Johnson Pharmaceutical Research and Development, Campus de Maigremont BP315, Val de Reuil, France, Virology Drug Discovery, Johnson & Johnson Pharmaceutical Research and Development, Tumhoutseweg 30 B-2340 Beerse, Belgium, TIBOTEC, General De Wittelaan L 11 B3, B-2800 Mechelen, Belgium, and Center for Advanced Biotechnology...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0408621

Reference43 articles.

1. Transmission of antiretroviral-drug-resistant HIV-1 variants

2. Adverse effects of antiretroviral therapy

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