Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V2 GPCR: Application To Ligand Screening and Oligomerization Assays.-Reference-Cited by-同舟云学术

Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V2 GPCR: Application To Ligand Screening and Oligomerization Assays.

Published:2012-10-05 Issue:20 Volume:55 Page:8588-8602
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Loison Stéphanie¹,Cottet Martin²,Orcel Hélène²,Adihou Hélène¹,Rahmeh Rita²,Lamarque Laurent³,Trinquet Eric³,Kellenberger Esther¹,Hibert Marcel¹,Durroux Thierry²,Mouillac Bernard²,Bonnet Dominique¹

Affiliation:

1. Laboratoire d’Innovation Thérapeutique, UMR7200 CNRS/Université de Strasbourg, Faculté de Pharmacie, 74 route du Rhin, 67412 Illkirch, France

2. CNRS UMR 5203, INSERM U661, and Université Montpellier I et II, Institut de Génomique Fonctionnelle, Département de Pharmacologie Moléculaire, 141 rue de la Cardonille, 34094 Montpellier Cedex 5, France

3. Cisbio Bioassays, Parc Marcel Boiteux, BP84175, 30200 Codolet, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm3006146

Reference49 articles.

1. Drug Discovery: A Historical Perspective

2. Value of novelty?

3. Fluorescence techniques: shedding light on ligand–receptor interactions

4. Fluorescence Polarization and Anisotropy in High Throughput Screening: Perspectives and Primer

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