Fluorescent Derivatives of AC-42 To Probe Bitopic Orthosteric/Allosteric Binding Mechanisms on Muscarinic M1 Receptors-Reference-Cited by-同舟云学术

Fluorescent Derivatives of AC-42 To Probe Bitopic Orthosteric/Allosteric Binding Mechanisms on Muscarinic M1 Receptors

Published:2012-02-27 Issue:5 Volume:55 Page:2125-2143
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Daval Sandrine B.¹,Valant Céline²,Bonnet Dominique²,Kellenberger Esther²,Hibert Marcel²,Galzi Jean-Luc¹,Ilien Brigitte¹

Affiliation:

1. Unité Biotechnologie et Signalisation Cellulaire, UMR 7242 CNRS, Ecole Supérieure de Biotechnologie de Strasbourg, Université de Strasbourg, BP 10413, 67412 Illkirch, France

2. Laboratoire d’Innovation Thérapeutique, UMR 7200 CNRS, Faculté de Pharmacie, Université de Strasbourg, 74 Route du Rhin, BP 24, 67401 Illkirch, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201348t

Reference62 articles.

1. Muscarinic Receptor Subtype Pharmacology and Physiology

2. Muscarinic acetylcholine receptors: mutant mice provide new insights for drug development

3. Allosteric activators of muscarinic receptors as novel approaches for treatment of CNS disorders

4. Allosterism at Muscarinic Receptors: Ligands and Mechanisms

5. Allosteric ligands for G protein-coupled receptors: A novel strategy with attractive therapeutic opportunities

Cited by 37 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Allosteric Modulation of Ligand Binding to Muscarinic Receptors;Neuromethods;2024

2. Investigation of Muscarinic Receptors by Fluorescent Techniques;Neuromethods;2024

3. Exploring Muscarinic Acetylcholine Receptor Binding Kinetics with Fluorescence Anisotropy;Neuromethods;2024

4. Designing drugs and chemical probes with the dualsteric approach;Chemical Society Reviews;2023

5. Multitargeting nature of muscarinic orthosteric agonists and antagonists;Frontiers in Physiology;2022-09-06