Enantiospecific Synthesis and Pharmacological Evaluation of a Series of Super-Potent, Conformationally Restricted 5-HT2A/2C Receptor Agonists-Reference-Cited by-同舟云学术

Enantiospecific Synthesis and Pharmacological Evaluation of a Series of Super-Potent, Conformationally Restricted 5-HT2A/2C Receptor Agonists

Published:2001-01-26 Issue:6 Volume:44 Page:1003-1010
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Chambers James J.¹,Kurrasch-Orbaugh Deborah M.¹,Parker Matthew A.¹,Nichols David E.¹

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, School of Pharmacy and Pharmacal Sciences, Purdue University, West Lafayette, Indiana 47907

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000491y

Reference24 articles.

1. Sanders-Bush, E.; Mayer, S. E. 5-Hydroxytryptamine (Serotonin) Receptor Agonists and Antagonists. InThe Pharmacological Basis ofTherapeutics, 9th ed.; Hardman, J. G., Limbird, L. E., Molinoff, P. B., Ruddon, R. W., Gilman, A. G., Eds.; McGraw-Hill: New York, 1996; pp 249−263.

2. Serotonin and Hallucinogens

3. Molecular biology of 5-HT receptors

4. Stereoselective LSD-like Activity in a Series of d-Lysergic Acid Amides of (R)- and (S)-2-Aminoalkanes

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