Effects of Amino Acid Chirality and the Chemical Linker on the Cell Permeation Characteristics of Cyclic Prodrugs of Opioid Peptides
Author:
Affiliation:
1. Department of Pharmaceutical Chemistry, The University of Kansas, Lawrence, Kansas 66047
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm050277f
Reference40 articles.
1. Improvement of oral peptide bioavailability: Peptidomimetics and prodrug strategies
2. BLOOD-BRAIN BARRIER DRUG TARGETING: THE FUTURE OF BRAIN DRUG DEVELOPMENT
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4. Structural requirements for intestinal absorption of peptide drugs
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