Design and Optimization of Benzimidazole-Containing Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists-Reference-Cited by-同舟云学术

Design and Optimization of Benzimidazole-Containing Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

Published:2010-12-03 Issue:1 Volume:54 Page:233-247
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Parks Daniel J.¹,Parsons William H.¹,Colburn Raymond W.¹,Meegalla Sanath K.¹,Ballentine Shelley K.¹,Illig Carl R.¹,Qin Ning¹,Liu Yi¹,Hutchinson Tasha L.¹,Lubin Mary Lou¹,Stone Dennis J.¹,Baker Judith F.¹,Schneider Craig R.¹,Ma Jianya¹,Damiano Bruce P.¹,Flores Christopher M.¹,Player Mark R.¹

Affiliation:

1. Janssen Research and Development, Welsh and McKean Roads, Spring House, Pennsylvania 19477-0776, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm101075v

Reference40 articles.

1. Identification of a cold receptor reveals a general role for TRP channels in thermosensation

2. A TRP Channel that Senses Cold Stimuli and Menthol

3. Inhibition of TRPM8 by Icilin Distinct from Desensitization Induced by Menthol and Menthol Derivatives

4. Tissue Distribution Profiles of the Human TRPM Cation Channel Family

Cited by 59 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Mechanisms of sensory adaptation and inhibition of the cold and menthol receptor TRPM8;Science Advances;2024-08-02

2. Subcutaneous administration of a novel TRPM8 antagonist reverses cold hypersensitivity while attenuating the drop in core body temperature;British Journal of Pharmacology;2024-05-24

3. Benzalkonium chloride, a common ophthalmic preservative, compromises rat corneal cold sensitive nerve activity;The Ocular Surface;2022-10

4. Transient Receptor Potential Channels: Important Players in Ocular Pain and Dry Eye Disease;Pharmaceutics;2022-09-02

5. Concise Synthesis of 7-Deoxypsammaplysins K and O and 7-Deoxyceratinamide A by 1,3-Dipole Cycloaddition;Organic Letters;2022-05-23