Aminopyrazole–Phenylalanine Based GPR142 Agonists: Discovery of Tool Compound and in Vivo Efficacy Studies-Reference-Cited by-同舟云学术

Aminopyrazole–Phenylalanine Based GPR142 Agonists: Discovery of Tool Compound and in Vivo Efficacy Studies

Published:2013-06-03 Issue:9 Volume:4 Page:829-834
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Yu Ming¹,Lizarzaburu Mike¹,Motani Alykhan¹,Fu Zice¹,Du Xiaohui¹,Liu Jiwen (Jim)¹,Jiao Xianyun¹,Lai SuJen¹,Fan Peter¹,Fu Angela¹,Liu Qingxiang¹,Murakoshi Michiko²,Nara Futoshi²,Oda Kozo²,Okuyama Ryo²,Reagan Jeff D.¹,Watanabe Nobuaki²,Yamazaki Mami²,Xiong Yumei¹,Zhang Ying¹,Zhuang Run¹,Lin Daniel C.-H.¹,Houze Jonathan B.¹,Medina Julio C.¹,Li Leping¹

Affiliation:

1. Amgen Inc., 1120 Veterans Boulevard, South San Francisco, California 94080, United States

2. Daiichi-Sankyo, 1-2-58 Hiromachi, Shinagawa-Ku, Tokyo 140-8710; 1-16-13 Kitakasai, Edogawa-Ku, Tokyo 134-8650, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml4000854

Reference5 articles.

1. Seven evolutionarily conserved human rhodopsin G protein-coupled receptors lacking close relatives

2. Characterisation and differential expression of two very closely related G-protein-coupled receptors, GPR139 and GPR142, in mouse tissue and during mouse development