Design, Synthesis, and Protein Crystallography of Biaryltriazoles as Potent Tautomerase Inhibitors of Macrophage Migration Inhibitory Factor
Author:
Affiliation:
1. Department of Chemistry, Yale University, New Haven, Connecticut 06520-8107, United States
Funder
National Institute of General Medical Sciences
Division of Graduate Education
Yale University
Debiopharm S.A.
Publisher
American Chemical Society (ACS)
Subject
Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis
Link
https://pubs.acs.org/doi/pdf/10.1021/ja512112j
Reference39 articles.
1. MIF: a new cytokine link between rheumatoid arthritis and atherosclerosis
2. Autoimmune diseases: MIF as a therapeutic target
3. The vascular biology of macrophage migration inhibitory factor (MIF)
4. Inflammation and cancer: macrophage migration inhibitory factor (MIF)--the potential missing link
5. Targeting the heat shock protein 90
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