Imidazolopiperazines: Lead Optimization of the Second-Generation Antimalarial Agents-Reference-Cited by-同舟云学术

Imidazolopiperazines: Lead Optimization of the Second-Generation Antimalarial Agents

Published:2012-04-23 Issue:9 Volume:55 Page:4244-4273
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nagle Advait¹,Wu Tao¹,Kuhen Kelli¹,Gagaring Kerstin¹,Borboa Rachel¹,Francek Caroline¹,Chen Zhong¹,Plouffe David¹,Lin Xuena²,Caldwell Christopher²,Ek Jared¹,Skolnik Suzanne²,Liu Fenghua²,Wang Jianling²,Chang Jonathan¹,Li Chun¹,Liu Bo¹,Hollenbeck Thomas¹,Tuntland Tove¹,Isbell John¹,Chuan Tiffany¹,Alper Philip B.¹,Fischli Christoph³⁴,Brun Reto³⁴,Lakshminarayana Suresh B.⁵,Rottmann Matthias³⁴,Diagana Thierry T.⁵,Winzeler Elizabeth A.¹,Glynne Richard¹,Tully David C.¹,Chatterjee Arnab K.¹

Affiliation:

1. Genomics Institute of the Novartis Research Foundation, 10675 John Jay Hopkins Drive, San Diego, California 92121, United States

2. Novartis Institute for Biomedical Research, Preclinical Profiling Group, Cambridge, Massachusetts

3. Swiss Tropical and Public Health Institute, Parasite Chemotherapy, CH-4002 Socinstrasse 57, CD-4002 Basel, Switzerland

4. University of Basel, CH-4003 Basel, Switzerland

5. Novartis Institute for Tropical Diseases, 10 Biopolis Road, 05-01 Chromos, Singapore-138670

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300041e

Reference28 articles.

1. Spiroindolones, a Potent Compound Class for the Treatment of Malaria

2. Road Towards New Antimalarials – Overview of the Strategies and their Chemical Progress

3. Evidence of Artemisinin-Resistant Malaria in Western Cambodia

4. The ‘Do Unto Others’ Malaria Vaccine

Cited by 91 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Ex vivo susceptibilities to ganaplacide and diversity in potential resistance mediators in Ugandan Plasmodium falciparum isolates;Antimicrobial Agents and Chemotherapy;2024-09-04

2. In vitro evaluation of ganaplacide/lumefantrine combination against Plasmodium falciparum in a context of artemisinin resistance;Journal of Antimicrobial Chemotherapy;2024-08-29

3. Synthesis of 4-morpholino-5,8,9,10-tetrahydropyrimido[4,5–b]quinolin-6(7H)-one derivatives and in silico-in vitro evaluation of their antimalarial activity;Results in Chemistry;2024-01

4. Key Contributions by the Swiss Tropical and Public Health Institute Towards New and Better Drugs for Tropical Diseases;CHIMIA;2023-09-20

5. Convenient Approach to 10‐ and 11‐Membered Azalactams;European Journal of Organic Chemistry;2023-04-17