Synthesis and Structure−Activity Relationships of Carboxylated Chalcones: A Novel Series of CysLT1 (LTD4) Receptor Antagonists-Reference-Cited by-同舟云学术

Synthesis and Structure−Activity Relationships of Carboxylated Chalcones: A Novel Series of CysLT1 (LTD4) Receptor Antagonists

Published:1997-03-01 Issue:7 Volume:40 Page:1075-1089
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zwaagstra Mariël E.¹,Timmerman Hendrik¹,Tamura Masahiro¹,Tohma Tsutomu¹,Wada Yasushi¹,Onogi Kazuhiro¹,Zhang Ming-Qiang¹

Affiliation:

1. Leiden/Amsterdam Centre for Drug Research, Division of Medicinal Chemistry, Vrije Universiteit, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands, and Tokyo Research Laboratories, Pharmaceutical Division, Kowa Company Ltd., 2-17-43, Tokyo Research Laboratories, Noguchi-Cho, Higashimurayama, Tokyo 189, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960628d

Reference54 articles.

1. Leukotrienes: Biosynthesis, Metabolism, and Pathophysiologic Significance

2. Leukotriene receptor antagonists and biosynthesis inhibitors: potential breakthrough in asthma therapy

3. Cysteinyl Leukotriene Production in Anaphylactic Reactions

4. Leukotrienes as a Target in Asthma Therapy

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