10-Ketomorphinan and 3-Substituted-3-desoxymorphinan Analogues as Mixed κ and μ Opioid Ligands: Synthesis and Biological Evaluation of Their Binding Affinity at Opioid Receptors-Reference-Cited by-同舟云学术

10-Ketomorphinan and 3-Substituted-3-desoxymorphinan Analogues as Mixed κ and μ Opioid Ligands: Synthesis and Biological Evaluation of Their Binding Affinity at Opioid Receptors

Published:2003-12-09 Issue:1 Volume:47 Page:165-174
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zhang Ao¹,Xiong Wennan¹,Bidlack Jean M.¹,Hilbert James E.¹,Knapp Brian I.¹,Wentland Mark P.¹,Neumeyer John L.¹

Affiliation:

1. Alcohol and Drug Abuse Research Center, McLean Hospital, Harvard Medical School, 115 Mill Street, Belmont, Massachusetts 02478, Department of Pharmacology and Physiology, School of Medicine and Dentistry, University of Rochester, Rochester, New York 14642, and Department of Chemistry, Rensselaer Polytechnic Institute, Troy, New York 12180

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0304156

Reference41 articles.

1. (b) Fries, D. S. Opioid Analgesics.Foye'sPrinciples of Medicinal Chemistry; Williams, D. A.; Lemke, T. L., Lippincott Williams & Wilkins: Philadelphia, PA, 2002; pp 453−479.

2. Selective opioid receptor agonists and antagonists: research tools and potential therapeutic agents

3. κ-Opioid receptors and analgesia

Cited by 41 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Palliative Care and Cancer Pain;Pain Care Essentials and Innovations;2021

2. Novel Dimethyltyrosine–Tetrahydroisoquinoline Peptidomimetics with Aromatic Tetrahydroisoquinoline Substitutions Show in Vitro Kappa and Mu Opioid Receptor Agonism;ACS Chemical Neuroscience;2019-06-14

3. C-Homomorphinan Derivatives as Lead Compounds to Obtain Safer and More Clinically Useful Analgesics;Chemical and Pharmaceutical Bulletin;2017

4. Multitarget opioid ligands in pain relief: New players in an old game;European Journal of Medicinal Chemistry;2016-01

5. Levorphanol use: past, present and future;Postgraduate Medicine;2015-12-27