Kiloscale Buchwald–Hartwig Amination: Optimized Coupling of Base-Sensitive 6-Bromoisoquinoline-1-carbonitrile with (S)-3-Amino-2-methylpropan-1-ol-Reference-Cited by-同舟云学术

Kiloscale Buchwald–Hartwig Amination: Optimized Coupling of Base-Sensitive 6-Bromoisoquinoline-1-carbonitrile with (S)-3-Amino-2-methylpropan-1-ol

Published:2014-10-16 Issue:12 Volume:18 Page:1752-1758
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Sperry Jeffrey B.¹,Price Wiglesworth Kristin E.¹,Edmonds Ian²,Fiore Phillip²,Boyles David C.¹,Damon David B.¹,Dorow Roberta L.¹,Piatnitski Chekler Eugene L.³,Langille Jonathan³,Coe Jotham W.³

Affiliation:

1. Chemical Research and Development, Pfizer, Inc., 558 Eastern Point Road, Groton, Connecticut 06340, United States

2. Bridge Organics, 311 West Washington Street, Vicksburg, Michigan 49097, United States

3. Pfizer Worldwide Medicinal Chemistry, Pfizer, Inc., 558 Eastern Point Road, Groton, Connecticut 06340, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op5002319

Reference34 articles.

1. PALLADIUM-CATALYZED AROMATIC AMINATION OF ARYL BROMIDES WITHN,N-DI-ETHYLAMINO-TRIBUTYLTIN

2. Palladium-Catalyzed Aromatic Aminations with in situ Generated Aminostannanes

3. A Simple Catalytic Method for the Conversion of Aryl Bromides to Arylamines

4. Palladium-catalyzed formation of carbon-nitrogen bonds. Reaction intermediates and catalyst improvements in the hetero cross-coupling of aryl halides and tin amides

5. Palladium-catalyzed synthesis of arylamines from aryl halides. Mechanistic studies lead to coupling in the absence of tin reagents

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