Dimeric Zanamivir Conjugates with Various Linking Groups Are Potent, Long-Lasting Inhibitors of Influenza Neuraminidase Including H5N1 Avian Influenza-Reference-Cited by-同舟云学术

Dimeric Zanamivir Conjugates with Various Linking Groups Are Potent, Long-Lasting Inhibitors of Influenza Neuraminidase Including H5N1 Avian Influenza

Published:2005-03-16 Issue:8 Volume:48 Page:2964-2971
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Macdonald Simon J. F.¹,Cameron Rachel¹,Demaine Derek A.¹,Fenton Rob J.¹,Foster Graham¹,Gower David¹,Hamblin J. Nicole¹,Hamilton Stephanie¹,Hart Graham J.¹,Hill Alan P.¹,Inglis Graham G. A.¹,Jin Betty¹,Jones Haydn T.¹,McConnell Darryl B.¹,McKimm-Breschkin Jennifer¹,Mills Gail¹,Nguyen Van¹,Owens Ian J.¹,Parry Nigel¹,Shanahan Stephen E.¹,Smith Donna¹,Watson Keith G.¹,Wu Wen-Yang¹,Tucker Simon P.¹

Affiliation:

1. GlaxoSmithKline Medicines Research Centre, Gunnels Wood Road, Stevenage SG1 2NY, United Kingdom, Biota Holdings, Level 4, 616 St. Kilda Road, Melbourne, 3004, Victoria, Australia, and CSIRO Health Sciences and Nutrition, 343 Royal Parade Parkville, 3052, Victoria, Australia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm040891b

Reference18 articles.

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2. Reece, P. A.; Watson, K. G.; Wu, W.Y.; Jin, B.; Krippner, G. Y. PCT Int. Appl. WO 98/21243, 1998 (Chem. Abstr.1998,129, 28172).

3. Highly potent and long-acting trimeric and tetrameric inhibitors of influenza virus neuraminidase

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