Pharmacophore-Based Virtual Screening and Biological Evaluation of Small Molecule Inhibitors for Protein Arginine Methylation

Author:

Wang Juxian1,Chen Limin2,Sinha Sarmistha Halder1,Liang Zhongjie23,Chai Huifang4,Muniyan Sakthivel5,Chou Yu-Wei5,Yang Chao1,Yan Leilei1,Feng You1,Kathy Li Keqin6,Lin Ming-Fong5,Jiang Hualiang2,George Zheng Yujun1,Luo Cheng23

Affiliation:

1. Department of Chemistry, Program of Molecular Basis of Diseases, Georgia State University, P.O. Box 4098, Atlanta, Georgia 30302, United States

2. Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China

3. Center for Systems Biology, Soochow University, Jiangsu 215006, China

4. Department of Pharmacy, Guiyang College of Traditional Chinese Medicine, Guiyang 550002, China

5. Department of Biochemistry and Molecular Biology, University of Nebraska Medical Center, Omaha, Nebraska 68198, United States

6. State Key Laboratory of Medical Genomics, Shanghai Institute of Hematology, Rui Jin Hospital Affiliated to Shanghai Jiao Tong University School of Medicine, Shanghai, China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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