Discovery, Optimization, and Pharmacological Characterization of Novel Heteroaroylphenylureas Antagonists of C−C Chemokine Ligand 2 Function-Reference-Cited by-同舟云学术

Discovery, Optimization, and Pharmacological Characterization of Novel Heteroaroylphenylureas Antagonists of C−C Chemokine Ligand 2 Function

Published:2011-02-22 Issue:6 Volume:54 Page:1667-1681
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Laborde Edgardo¹,Macsata Robert W.¹,Meng Fanying¹,Peterson Brian T.¹,Robinson Louise¹,Schow Steve R.¹,Simon Reyna J.¹,Xu Hua¹,Baba Kunihisa²,Inagaki Hideaki²,Ishiwata Yoshiro²,Jomori Takahito²,Matsumoto Yukiharu²,Miyachi Atsushi²,Nakamura Takashi²,Okamoto Masayuki²,Handel Tracy M.³,Bernard Claude C. A.⁴

Affiliation:

1. Telik, Inc., 700 Hansen Way, Palo Alto, California 94304, United States

2. Sanwa Kagaku Kenkyusho Co., Ltd., Mie Research Park, 363 Shiosaki, Hokusei-Cho, Inabe-Shi, Mie, 511-0406, Japan

3. Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, 9500 Gilman Drive, La Jolla, California 92093, United States

4. Immunology and Stem Cell Laboratories, Monash University, Building 75, Wellington Road, Clayton, Victoria 3800, Australia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm1012903

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