Identification of Anxiolytic/Nonsedative Agents among Indol-3-ylglyoxylamides Acting as Functionally Selective Agonists at the γ-Aminobutyric Acid-A (GABAA) α2 Benzodiazepine Receptor-Reference-Cited by-同舟云学术

Identification of Anxiolytic/Nonsedative Agents among Indol-3-ylglyoxylamides Acting as Functionally Selective Agonists at the γ-Aminobutyric Acid-A (GABAA) α2 Benzodiazepine Receptor

Published:2009-05-26 Issue:12 Volume:52 Page:3723-3734
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Taliani Sabrina¹,Cosimelli Barbara¹,Da Settimo Federico¹,Marini Anna Maria¹,La Motta Concettina¹,Simorini Francesca¹,Salerno Silvia¹,Novellino Ettore¹,Greco Giovanni¹,Cosconati Sandro¹,Marinelli Luciana¹,Salvetti Francesca¹,L’Abbate Gianluca¹,Trasciatti Silvia¹,Montali Marina¹,Costa Barbara¹,Martini Claudia¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy, Dipartimento di Chimica Farmaceutica e Tossicologica, Università di Napoli “Federico II”, Via Domenico Montesano 49, 80131 Napoli, Italy, Abiogen Pharma SpA, Research Centre, Via del Paradiso 6, 56019 Migliarino Pisano, Pisa, Italy, Dipartimento di Psichiatria, Neurobiologia, Farmacologia e Biotecnologie, Università di Pisa, Via Bonanno 6, 56126 Pisa, Italy, Dipartimento di Morfologia Umana e Biologia Applicata,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9001154

Reference70 articles.

1. Mapping of the Benzodiazepine Recognition Site on GABA-A Receptors

2. GABA-Activated Ligand Gated Ion Channels: Medicinal Chemistry and Molecular Biology

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