Novel Octreotide Dicarba-analogues with High Affinity and Different Selectivity for Somatostatin Receptors-Reference-Cited by-同舟云学术

Novel Octreotide Dicarba-analogues with High Affinity and Different Selectivity for Somatostatin Receptors

Published:2010-07-28 Issue:16 Volume:53 Page:6188-6197
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Di Cianni Alessandra¹²,Carotenuto Alfonso³,Brancaccio Diego³,Novellino Ettore³,Reubi Jean Claude⁴,Beetschen Karin⁴,Papini Anna Maria¹²,Ginanneschi Mauro¹²

Affiliation:

1. Laboratory of Peptides & Proteins, Chemistry & Biology, University of Firenze, Via della Lastruccia 13, I-50019 Sesto Fiorentino, Italy

2. Department of Chemistry “Ugo Schiff”, University of Firenze, Via della Lastruccia 5-13, I-50019, Sesto Fiorentino, Italy

3. Department of Pharmaceutical Chemistry and Toxicology, University of Napoli, Via Domenico Montesano 49, I-80131 Napoli, Italy

4. Division of Cell Biology and Experimental Cancer Research, Institute of Pathology, University of Berne, Murtenstrasse 31, CH-3010 Berne, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm1005868

Reference49 articles.

1. Burgus, R.; Brazeau, P.; Vale, W. W.Isolation and determination of the primary structure of somatostatin (a somatotropin release inhibiting factor) of bovin hypothalamic origin.Advances in Human Growth Hormone Research, Report no. 74-612;U.S. Government Printing Office, DHEW, (NIH):Washington, DC, 1973; pp144−158.

2. Opportunities in somatostatin research: biological, chemical and therapeutic aspects

3. Novel, Potent, and Radio-Iodinatable Somatostatin Receptor 1 (sst1) Selective Analogues

4. Novel sst2-Selective Somatostatin Agonists. Three-Dimensional Consensus Structure by NMR

5. Conformational analysis of a potent SSTR3-selective somatostatin analogue by NMR in water solution

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