Potent, Selective, and Orally Efficacious Antagonists of Melanin-Concentrating Hormone Receptor 1-Reference-Cited by-同舟云学术

Potent, Selective, and Orally Efficacious Antagonists of Melanin-Concentrating Hormone Receptor 1

Published:2006-11-04 Issue:24 Volume:49 Page:7095-7107
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tavares Francis X.¹,Al-Barazanji Kamal A.¹,Bigham Eric C.¹,Bishop Michael J.¹,Britt Christy S.¹,Carlton David L.¹,Feldman Paul L.¹,Goetz Aaron S.¹,Grizzle Mary K.¹,Guo Yu C.¹,Handlon Anthony L.¹,Hertzog Donald L.¹,Ignar Diane M.¹,Lang Daniel G.¹,Ott Ronda J.¹,Peat Andrew J.¹,Zhou Hui-Qiang¹

Affiliation:

1. Department of Medicinal Chemistry, Department of Metabolic Diseases, Pharmaceutical Development, Department of Research Bioanalysis and Drug Metabolism, Discovery Research CASS, Department of Biochemical and Analytical Pharmacology, and Screening and Compound Profiling, GlaxoSmithKline, Research Triangle Park, North Carolina 27709

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060572f

Reference59 articles.

1. Characterization of melanin-concentrating hormone in chum salmon pituitaries

2. Characterization of Melanin-Concentrating Hormone from Rat Hypothalamus*

3. The melanin-concentrating hormone system of the rat brain: An immuno- and hybridization histochemical characterization

4. Melanin-concentrating hormone is the cognate ligand for the orphan G-protein-coupled receptor SLC-1

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