In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt1-DALDA Analogues-Reference-Cited by-同舟云学术

In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt1-DALDA Analogues

Published:2014-02-06 Issue:4 Volume:5 Page:352-357
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Ballet Steven¹,Betti Cecilia¹,Novoa Alexandre¹,Tömböly Csaba²,Uhd Nielsen Carsten³,Helms Hans Christian³,Lesniak Anna⁴,Kleczkowska Patrycja⁴,Chung Nga N.⁵,Lipkowski Andrzej W.⁴⁶,Brodin Birger³,Tourwé Dirk¹,Schiller Peter W.⁵

Affiliation:

1. Department of Organic Chemistry, Vrije Universiteit Brussel, Pleinlaan 2, B-1050 Brussels, Belgium

2. Laboratory of Chemical Biology, Biological Research Centre of the Hungarian Academy of Sciences, Temesvári, krt. 62, H-6726 Szeged, Hungary

3. The Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, 2100 Copenhagen, Denmark

4. Mossakowski Medical Research Centre Polish Academy of Sciences, Warsaw, Poland

5. Laboratory of Chemical Biology and Peptide Research, Clinical Research Institute of Montreal, Montreal, QC H2W 1R7, Canada

6. Tufts University School of Medicine, Boston, Massachusetts 02111, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml4004765

Reference28 articles.

1. Improved bioavailability to the brain of glycosylated Met-enkephalin analogs

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3. The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety

4. Opioid glycopeptide analgesics derived from endogenous enkephalins and endorphins

5. New glycosylpeptides with high antinociceptive activity

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