A 20S Combined with a 22R Configuration Markedly Increases both in Vivo and in Vitro Biological Activity of 1α,25-Dihydroxy-22-methyl-2-methylene-19-norvitamin D3-Reference-Cited by-同舟云学术

A 20S Combined with a 22R Configuration Markedly Increases both in Vivo and in Vitro Biological Activity of 1α,25-Dihydroxy-22-methyl-2-methylene-19-norvitamin D3

Published:2012-04-22 Issue:9 Volume:55 Page:4352-4366
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Flores Agnieszka¹,Sicinski Rafal R.²,Grzywacz Pawel¹,Thoden James B.¹,Plum Lori A.¹,Clagett-Dame Margaret¹,DeLuca Hector F.¹

Affiliation:

1. Department of Biochemistry, College of Agriculture and Life Sciences, University of Wisconsin-Madison, 433 Babcock Drive, Madison, Wisconsin 53706-1544, United States

2. Department of Chemistry, University of Warsaw, Pasteura 1, 02-093 Warsaw, Poland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300187x

Reference38 articles.

1. Current Understanding of the Molecular Actions of Vitamin D

2. Overview of general physiologic features and functions of vitamin D

3. A New Look at the Most Successful Prodrugs for Active Vitamin D (D Hormone): Alfacalcidol and Doxercalciferol

4. Vitamin D Analogs as Modulators of Vitamin D Receptor Action

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