Design and Synthesis of Novel Sulfonamide-Containing Bradykinin hB2 Receptor Antagonists. 1. Synthesis and SAR of α,α-Dimethylglycine Sulfonamides-Reference-Cited by-同舟云学术

Design and Synthesis of Novel Sulfonamide-Containing Bradykinin hB2 Receptor Antagonists. 1. Synthesis and SAR of α,α-Dimethylglycine Sulfonamides

Published:2006-05-20 Issue:12 Volume:49 Page:3602-3613
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Fattori Daniela¹,Rossi Cristina¹,Fincham Christopher I.¹,Berettoni Marco¹,Calvani Federico¹,Catrambone Fernando¹,Felicetti Patrizia¹,Gensini Martina¹,Terracciano Rosa¹,Altamura Maria¹,Bressan Alessandro¹,Giuliani Sandro¹,Maggi Carlo A.¹,Meini Stefania¹,Valenti Claudio¹,Quartara Laura¹

Affiliation:

1. Menarini Ricerche, Via Tito Speri 10, 00040 Pomezia (Roma), Italy, and Menarini Ricerche, Via Rismondo 12A, Firenze, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060137l

Reference34 articles.

1. MEN16132, a novel potent and selective nonpeptide antagonist for the human bradykinin B2 receptor. In vitro pharmacology and molecular characterization

2. Bradykinin receptors: Pharmacological properties and biological roles

3. Biochemical and Molecular Pharmacology of Kinin Receptors

4. Cloning and pharmacological characterization of a human bradykinin (BK-2) receptor

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