Synthesis of Nitroindole Derivatives with High Affinity and Selectivity for Melatoninergic Binding Sites MT3-Reference-Cited by-同舟云学术

Synthesis of Nitroindole Derivatives with High Affinity and Selectivity for Melatoninergic Binding Sites MT3

Published:2002-03-27 Issue:9 Volume:45 Page:1853-1859
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Leclerc Véronique¹,Yous Saïd¹,Delagrange Philippe¹,Boutin Jean A.¹,Renard Pierre¹,Lesieur Daniel¹

Affiliation:

1. Institut de Chimie Pharmaceutique Albert Lespagnol, 3 rue du Professeur Laguesse, BP83, 59006 Lille Cedex, France, Institut de Recherches Internationales Servier, 1 rue Carle Hébert, 92415 Courbevoie Cedex, France, and Division de Pharmacologie Moléculaire et Cellulaire, Institut de Recherches Servier, 125 Chemin de Ronde, 78290 Croissy-sur-Seine, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm011053%2B

Reference26 articles.

1. Pineal Melatonin: Cell Biology of Its Synthesis and of Its Physiological Interactions*

2. Melatonin receptors: Localization, molecular pharmacology and physiological significance

3. Melatonin, Its Receptors, and Relationships with Biological Rhythm Disorders

4. Expression cloning of a high-affinity melatonin receptor from Xenopus dermal melanophores.

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