1. Medicinal Chemistry, Department of Pharmacy and Pharmacology and Sterix Ltd., University of Bath, Claverton Down, Bath, BA2 7AY, United Kingdom, Dipartimento di Scienze Biomediche e Biotecnologie, Università di Brescia, Viale Europa 11, 25133 Brescia, Italy, JASCO Corporation, 2967-5 Ishikawa-cho, Hachioji-shi, Tokyo, Japan, Endocrinology and Metabolic Medicine and Sterix Ltd., Imperial College London, Faculty of Medicine, St. Mary’s Hospital, London, W2 1NY, United Kingdom