Selectivity and Mechanism of Action of a Growth Factor Receptor-Bound Protein 2 Src Homology 2 Domain Binding Antagonist-Reference-Cited by-同舟云学术

Selectivity and Mechanism of Action of a Growth Factor Receptor-Bound Protein 2 Src Homology 2 Domain Binding Antagonist

Published:2008-11-07 Issue:23 Volume:51 Page:7459-7468
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Giubellino Alessio¹,Shi Zhen-Dan¹,Jenkins Lisa M. Miller¹,Worthy Karen M.¹,Bindu Lakshman K.¹,Athauda Gagani¹,Peruzzi Benedetta¹,Fisher Robert J.¹,Appella Ettore¹,Burke Terrence R.¹,Bottaro Donald P.¹

Affiliation:

1. Urologic Oncology Branch and Laboratory of Cell Biology, National Cancer Institute, Bethesda, Maryland 20892, Laboratory of Medicinal Chemistry, National Cancer Institute at Frederick, Frederick, Maryland 21702 and Protein Chemistry Laboratory-SAIC, Frederick, Maryland 21702

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800523u

Reference28 articles.

1. Oncogenic kinase signalling

2. The SH2 and SH3 domain-containing protein GRB2 links receptor tyrosine kinases to ras signaling

3. GRB2: A pivotal protein in signal transduction

4. p21-activated kinases in cancer

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